Cleavable linkers in antibody–drug conjugates
Accepted version
Peer-reviewed
Repository URI
Repository DOI
Change log
Authors
Bargh, Jonathan D
Isidro-Llobet, Albert
Parker, Jeremy S
Spring, David R
Abstract
This tutorial review summarises the advances in the field of cleavable linker technologies for antibody–drug conjugates (ADCs).
Description
Keywords
Acids, Animals, Antibodies, Monoclonal, Antineoplastic Agents, Cathepsin B, Disulfides, Drug Stability, Humans, Immunoconjugates
Journal Title
Chemical Society Reviews
Conference Name
Journal ISSN
0306-0012
1460-4744
1460-4744
Volume Title
Publisher
Royal Society of Chemistry (RSC)
Publisher DOI
Sponsorship
Engineering and Physical Sciences Research Council (1800455)